Gloria Maria da Silva, Daniel Henrique Berto de Souza, Karoline B. Waitman, Matteo Celano Ebram, Melissa R. Fessel, Iuliu Cezar Zainescu, Fernanda C. Portaro, Montse Heras, Sonia A. de Andrade* "Design, synthesis, and evaluation of Bothrops venom serine protease peptidic inhibitors." Journal Of Venomous Animals And Toxins Including Tropical Diseases 27 (2021): 1-7. Belo RF, Martins MLF; Shvachiy L; Costa-Coelho T; de Almeida-Borlido C; Fonseca-Gomes J; Neves V; Vicente Miranda H, Outeiro TF; Coelho JE, Xapelli S, Valente CA; Heras M; Bardaji E; Castanho MARB; Diogenes MJ; Sebastião AM "The Neuroprotective Action of Amidated-Kyotorphin on Amyloid &b. Peptide Induced Alzheimer's Disease Pathophysiology." Frontiers in Pharmacology 11 (2020): -. Vitor Martins de Andrade, Eduard Bardají, Montserrat Heras, Vasanthakumar G. Ramu, Juliana Campos Junqueira, Jéssica Diane dos Santos, Miguel A.R.B. Castanho, Katia Conceiçao "Antifungal and anti-biofilm activity of designed derivatives from kyotorphin." Fungal Biology (2019): -. Juliana Perazzo; Carla Lima; Montserrat Heras; Eduard Bardají; Mônica Lopes-Ferreira; Miguel Castanho "Neuropeptide kyotorphin impacts on lipopolysaccharide-induced glucocorticoid-mediated inflammatory response. A molecular link to nociception, neuroprotection, and anti-Inflammatory action." ACS Chemical Neuroscience 8 (2017): -. Figueira, T. N.; Freire, J. M.; Cunha-Santos, C.; Heras, M.; Gonçalves, J.; Moscona, A.; Porotto, M.; Veiga, A. S.; Castanho, M. A. R. B. "Quantitative analysis of molecular partition towards lipid membranes using surface plasmon resonance." Scientific Reports 7 (2017): art.45647-. Juliana Perazzo; Mônica Lopes-Ferreira; Sónia Sá Santos; Isa Serrano; Antónia Pinto; Carla Lima; Eduard Bardaji; Isaura Tavares; Montserrat Heras; Katia Conceição; Miguel A. R. B. Castanho "Endothelium-Mediated action of analogues of the endogenous neuropeptide kyotorphin (Tyrosil-Arginine): mechanistic insights from permeation and effects on microcirculation." ACS Chemical Neuroscience 7 (2016): 1130-1140. Maria Cristina Oliveira; Lurdes Gano; Isabel Santos; João D. G. Correia; Isa D. Serrano; Sónia Sá Santos; Marta Ribeiro; Juliana Perazzo; Isaura Tavares; Montserrat Heras; Eduard Bardaji; Miguel A. Castanhob "Improvement of the pharmacological properties of amidated kyotorphin by means of iodination." MedChemComm 7 (2016): 906-913. Santos, Sónia Sá; Santos, Sara Matos; Pinto, Antónia R T; Ramu, Vasanthakumar Ganga; Heras i Corominas, Montserrat; Bardají Rodríguez, Eduard; Tavares, Isaura R.; and Castanho, Miguel Augusto Rico Botas "Amidated and ibuprofen-conjugated kyotorphins promote neuronal rescue and memory recovery in cerebral hypoperfusion dementia model." Frontiers in Aging Neuroscience 8 (2016): 1-11. Conceição, Katia; Magalhães, Pedro R.; Campos, Sara R R; Domingues, Marco M.; Ramu, Vasanthakumar G.; Michalek, Matthias; Bertani, Philippe; Baptista, António M.; Heras, Montserrat; Bardají Rodríguez, Eduard; Bechinger, Burkh "The Anti‑inflammatory action of the analgesic kyotorphin neuropeptide derivatives: insights of a lipid‑mediated mechanism." Amino Acids 48 (2016): 307-318. El Marrouni El Ghazaoui, Abdellatif ; Heras i Corominas, Montserrat "Synthesis of new unnatural Nα-Fmoc pyrimidin-4-one amino acids: use of the p-benzyloxybenzyloxy group as a pyrimidinone masking group." Organic and Biomolecular Chemistry 13 (2015): 851-858. Serrano, Isa D.; Ramu, Vasanthakumar Ganga; Pinto, Antónia R T; Freire, João M.; Tavares, Isaura R.; Heras i Corominas, Montserrat; Bardají Rodríguez, Eduard; Castanho, Miguel Augusto Rico Botas "Correlation Between Membrane Translocation and Analgesic Efficacy in Kyotorphin Derivatives." Biopolymers (títol associat amb Peptide Science) 104 (2015): 1-10. Vasanthakumar G. Ramu; Eduard Bardaji; Montserrat Heras "DEPBT coupling reagent avoid racemization in solution phase synthesis of a kyotorphin derivative." Synthesis : journal of synthetic organic chemistry 46 (2014): 1481-1486. Abdelatif ElMarrouni; Amandine Kolleth; Raphael Lebeuf; Julian Gebauer; Sébastien Prevost; Montserrat Heras, Stellios Arseniyadis; Janine Cossy "Lyngbouilloside and Related Macrolides from Marine Cyanobacteria." Natural Product Communications 8 (2013): 965-972. Marta M.B. Ribeiro; Sónia Sá Santos; David S. C. Sousa; Margarita Oliveira; Sara M. Santos; Montserrat Heras; Eduard R. Bardaji; Isaura Tavares; Miguel A.R.B. Castanho "Side-effects of analgesic Kyotorphin derivatives: advantages over clinical opioid drugs." Amino Acids 45 (2013): 171-178. Marta M.B. Ribeiro; Henri G. Franquelim; Inês M. Torcato; Vasanthakumar G. Ramu; Montserrat Heras; Eduard R. Bardaji; Miguel A.R.B. Castanho "Antimicrobial properties of analgesic kyotorphin peptides unraveled through atomic force microscopy." Biochemical and Biophysical Research Communications 420 (2012): 676-679. ElMarrouni, A.; Lebeuf, R.; Gebauer, J.; Heras, M.; Arseniyadis, S.; Cossy, J. "Total synthesis of nominal Lyngbouilloside aglycon." Organic Letters 14 (2012): 314-317. ElMarrouni, A.; Fabrellas, J.; Heras, M. "Coupling reaction between electron-rich pyrimidinones and alpha-amino acids promoted by phosphonium salts." Organic and Biomolecular Chemistry 9 (2011): 5967-5977. Ribeiro, M.M.M.; Pinto, A.; Pinto, M.; Heras, M.; Martins, I.; Correia, A. Bardají, E.; Tavares, I.; Castanho, M. "Inhibition of nociceptive responses after systemic administration of amidated kyotorphin." British Journal of Pharmacology 163 (2011): 964-973. Ribeiro, M.M.M.; Pinto, A.; Domingues, M. M.; Serrano, I.; Heras, M.; Bardají, E.; Tavares, I.; Castanho, M. "Chemical conjugation of neuropeptide kyotorphin and ibuprofen enhaces brain targeting and analgesis." Molecular Pharmaceutics 8 (2011): 1929-1940. Elmarrouni, A.; Shyamsunder R. Joolakanti; Colon, A.; Heras, M.; Arseniyadis, S.; Cossy, J. "Two concise total syntheses of (-)-bitungolide F." Organic Letters 12 (2010): 4074-4077. Elmarrouni, A.; Fukuda, A.; Heras, M.; Arseniyadis, S.; Cossy, J. "Expedient synthesis of a stereoisomer of acremolide B." Journal of Organic Chemistry 75 (2010): 8478-8486. Elmarrouni, A.; Güell, M.; Collell, C.; Heras, M. "A Simple approach for the synthesis of new pyrimidinyl alpha-amino acids." Tetrahedron 66 (2010): 612-623. Font, D.; Heras, M.; Villalgordo, J.M. "Synthesis of pyrimidinyl arylglycines through subsequent Mitsunobu and Petasis reactions." Tetrahedron 64 (2008): 5226-5235. Font, D. ; Linden, A. ; Heras, M. ; Villalgordo, J. M. "A simple approach for the regioselective synthesis of imidazo[1,2-a]pyrimidinones and pyrimido[1,2-a]pyrimidinones." Tetrahedron 62 (2006): 1433-1443. Heras, M.; Gulea M.; Masson, S.; Philouze, C. "A Hetero-Diels-Alder Approach to Phosphonothiashikimc Acid and New Thiaglycosides." European Journal of Organic Chemistry 2004 (2004): 160-172. Heras, M.; Font, D.; Linden, A.; Villalgordo, J.M. "Synthesis of triazolo[1,5-a]triazin-7-one derivatives and highly functionalized [1,2,4]triazoles." Helvetica Chimica Acta 86 (2003): 3204-3214. Font, D.; Heras, M.; Villalgordo, J.M. "Solution- and solid-phase parallel synthesis of 4-alkoxy-substituted pyrimidines with high molecular diversity Synthesis of 4-Alkoxy-Substituted Pyrimidines with High Molecular Diversity." Journal of Combinatorial Chemistry 5 (2003): 311-321. Font, D.; Heras, M.; Villalgordo, J.M. "Development of an efficient and straightforward methodology toward the synthesis of molecularly diverse 2,6-disubstituted 3,4-dihydropyrimidin-4(3H)-ones." Synthesis : journal of synthetic organic chemistry (2002): 1833-1843. Moreno, P.; Heras, M.; Maestro, M.; Villalgordo, J.M. "Synthesis of novel 2,3-dihydroimidazo[2,1b][1,3] oxazoles through intramolecular nucleophilic ipso-substitution in 2-alkysulfonylimidazoles." Synthesis : journal of synthetic organic chemistry (2002): 2691-2700. Heras, M.; Ventura, M.; Linden, A.; Villalgordo, J.M. "Reaction of α-iminomethylene amino esters with mono- and bidentate nucleophiles: a straightforward route to 2-amino-1H-5-imidazolones." Tetrahedron 57 (2001): 4371-4388. Heras, M.; Gulea, M.; Masson, S. "First synthesis of a phosphonothiashikimic acid derivative." Chemical Communications 2001 (2001): 611-612. Heuzé, B.; Gasparova, R.; Heras, M.; Masson, S. "Phosphonodithioformates as heterodienophiles: synthesis of (3,6-dihydro-2H-thiopyran-2-yl)phosphonates." Tetrahedron Letters 41 (2000): 7327-7331. Heras M., Ventura M., Linden A., Villalgordo J.M. "Intramolecular Nucleophilic ipso-Substitution in 2-Alkylsulfonylimidazoles Produces New Class of Fused Imidazoles: Síntesis of 2,3-Dihydroimidazo[2,1-b][1,3] Oxazoles." Synthesis : journal of synthetic organic chemistry (1999): 1613-1624. Heras, M.; Planas, M.; Rafel, S.; Ventura, M.; Ortuño R. M. "Synthesis of new polyfunctional 1-oxaspiro [4.4]nonanes and 1-oxaspiro [4.5]decanes: a general methodology." Anales de Quimica-International Edition (1996): 233-242.